CAS:574013-66-4 | Fexaramine

Introduction and application of CAS:574013-66-4 | Fexaramine

Fexaramine is a potent and selective farnesoidXreceptor (FXR) agonist with an EC50 of 25nM. It is inactive against hRXRα, hPPARα, hPPARγ, hPPARδ, mPXR, hPXR, hLXRα, hTRβ, hRARβ, mCAR, mERRγ and hVDR receptors.

Specification of CAS:574013-66-4 | Fexaramine

Boiling point: 677.7±55.0°C(Predicted)
Density: 1.158±0.06g/cm3(Predicted)
Storage conditions: 2-8°C
Solubility: DMSO: 50mg/mL (100.68mM; ultrasound required)
Form: powder
Acidity coefficient (pKa): 4.95±0.24 (Predicted)
color: White

Package and transportation of CAS:574013-66-4 | Fexaramine

Transportation: by courier/ by air/ by sea.

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